Список публикаций Лаборатории синтеза антибиотиков, преодолевающих резистентность (САПР)

 

  1. I.B. Levshin, A.Y. Simonov, A.A. Panov, N.E. Grammatikova, A.I. Alexandrov, E.S.M.O. Ghazy, V.A. Ivlev, M.O. Agaphonov, A.B. Mantsyzov, V.I. Polshakov, Synthesis and Biological Evaluation of a Series of New Hybrid Amide Derivatives of Triazole and Thiazolidine-2,4-dione, Pharmaceuticals, 2024, 17, 723; https://doi.org/10.3390
    /ph17060723

  2. A.A. Panov, New Methods of Synthesis of Fused Maleimides, Russian Journal of Organic Chemistry, 2024, 60, 553–567; https://doi.org/10.1134/S1070428024040018
     

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  3. D.V. Andreeva, A.S. Tikhomirov, A.E. Shchekotikhin, Synthesis and antiproliferative activity of thiazole-fused anthraquinones, Organic & Biomolecular Chemistry, 2024, in press; https://doi.org/10.1039/D4OB01284D 
     

  4. V.N. Charushin, E.V. Verbitskiy, O.N. Chupakhin, D.V. Vorobyeva, P.S. Gribanov, S.N. Osipov, A.V. Ivanov, S.V. Martynovskaya, E.F. Sagitova, V.D. Dyachenko, I.V. Dyachenko, S.G. Krivokolysko, V.V. Dotsenko, A.V. Aksenov, D.A. Aksenov, N.A. Aksenov, A.A. Larin, L.L. Fershtat, V.M. Muzalevskiy, V.G. Nenajdenko, A.V. Gulevskaya, A.F. Pozharskii, E.A. Filatova, K.V. Belyaeva, B.A. Trofimov, I.A. Balova, N.A. Danilkina, A.I. Govdi, A.S. Tikhomirov, A.E. Shchekotikhin, M.S. Novikov, N.V. Rostovskii, A.F. Khlebnikov, Yu.N. Klimochkin, M.V. Leonova, I.M. Tkachenko, V.A. Mamedov, V.L. Mamedova, N.A. Zhukova, V.E. Semenov, O.G. Sinyashin, O.V. Borshchev, Yu.N. Luponosov, S.A. Ponomarenko, A.S. Fisyuk, A.S. Kostyuchenko, V.G. Ilkin, T.V. Beryozkina, V.A. Bakulev, A.S. Gazizov, A.A. Zagidullin, A.A. Karasik, M.E. Kukushkin, E.K. Beloglazkina, N.E. Golantsov, A.A. Festa, L.G. Voskresensky, V.S. Moshkin, E.M. Buev, V.Ya. Sosnovskikh, I.A. Mironova, P.S. Postnikov, V.V. Zhdankin, M.S. Yusubov, I.A. Yaremenko, V.A. Vil', I.B. Krylov, A.O. Terent'ev, Yu.G. Gorbunova, A.G. Martynov, A.Yu. Tsivadze, P.A. Stuzhin, S.S. Ivanova, O.I. Koifman, O.N. Burov, M.E. Kletskii, S.V. Kurbatov, O.I. Yarovaya, K.P. Volcho, N.F. Salakhutdinov, M.A. Panova, Ya.V. Burgart, V.I. Saloutin, A.R. Sitdikova, E.S. Shchegravina, A.Yu. Fedorov, The chemistry of heterocycles in the 21st century, Russian Chemical Reviews, 2024, 93 (7), RCR5125; https://doi.org/10.59761/RCR5125
     

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  5. D.V. Andreeva, T.S. Vedekhina, A.S. Gostev, L.G. Dezhenkova, Y.L. Volodina, A.A. Markova, M.T. Nguyen, O.M. Ivanova, V.A. Dolgusheva, A.M. Varizhuk, A.S. Tikhomirov, A.E. Shchekotikhin, Thiadiazole-, selenadiazole- and triazole-fused anthraquinones as G-quadruplex targeting anticancer compounds, European Journal of Medicinal Chemistry, 2024, 268, 116222; https://doi.org/10.1016/j.ejmech.2024.116222

  6. I.A. Volynkina, E.N. Bychkova, A.O. Karakchieva, A.S. Tikhomirov, G.V. Zatonsky, S.E. Solovieva, M.M. Martynov, N.E. Grammatikova, A.G. Tereshchenkov, A. Paleskava, A.L. Konevega, P.V. Sergiev, O.A. Dontsova, I.A. Osterman, A.E. Shchekotikhin, A.N. Tevyashova, Hybrid Molecules of Azithromycin with Chloramphenicol and Metronidazole: Synthesis and Study of Antibacterial Properties, Pharmaceuticals, 2024, 17 (2), 187; https://doi.org/10.3390/ph17020187

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  7. V.A.Litvinova, A.S.Tikhomirov, A.E.Shchekotikhin, Methods for functionalization of anthraquinones, Russian Chemical Reviews, 2024, 93, RCR5141, DOI: https://doi.org/10.59761/RCR5141

  8. A.S. Tikhomirov, Y.B. Sinkevich, L.G. Dezhenkova, D.N. Kaluzhny, N.S. Ilyinsky, V.I. Borshchevskiy, D. Schols, A.E. Shchekotikhin, Synthesis and antitumor activity of cyclopentane-fused anthraquinone derivatives, European Journal of Medicinal Chemistry, 2024, 265, 116103, https://doi.org/10.1016/j.ejmech.2023.1161031
  9. M.I. Treshchalin, V.A. Polozkova, E.I. Moiseenko, A.E. Shchekotikhin, S.A. Dovzhenko, M.B. Kobrin, E.R. Pereverzeva, Experimental Evaluation of the Hypersensitivity Reactions of a New Glycopeptide Antibiotic Flavancin in Animal Models, Pharmaceuticals, 2023, 16(11), 1569; https://doi.org/10.3390/ph16111569 img

     

  10. V.A. Litvinova, A.S. Gostev, A.S. Tikhomirov, A.E. Shchekotikhin, New heteroarene-fused anthraquinones: Synthesis and PyBOP-mediated amination, Tetrahedron, 2023, 149, 4, 133722, https://doi.org/https://doi.org/10.1016/j.tet.2023.133722img

     

  11. A. Islam, X.C. Chen, C.-W. Weng, C.-Y. Chen, C.-W. Wang, M.-K. Chen, A.S. Tikhomirov, A.E. Shchekotikhin, P.J. Chueh, Water-soluble 4-(dimethylaminomethyl)heliomycin exerts greater antitumor effects than parental heliomycin by targeting the tNOX-SIRT1 axis and apoptosis in oral cancer cells, eLife, 2023, https://doi.org/10.7554/eLife.87873.1img

     

  12. В.А. Литвинова, А.С. Тихомиров, Методы синтеза 1,3-оксазолидин-2-онов, Методы синтеза 1,3-оксазолидин-2-онов, Химия гетероциклических соединений, 2023, 59(11/12), 733-735img

     

  13. K. Shapovalova, G. Zatonsky, N. Grammatikova, I. Osterman, E. Razumova, A. Shchekotikhin, A. Tevyashova, Synthesis of 6”-Modified Kanamycin A Derivatives and Evaluation of Their Antibacterial Properties. Pharmaceutics, 2023, 15, 1177. https://doi.org/10.3390/pharmaceutics15041177img

     

  14. A.A. Panov, Quantum-Chemical Study of Keto-Enol Equilibrium and Global Electrophilicity of Hydroxymaleimide Derivatives. Doklady Physical Chemistry, 2023, 508, 28–32, https://doi.org/10.1134/S001250162360002Ximg

     

  15. Levshin I.B., Simonov A.Y., Lavrenov S.N., Panov A.A., Grammatikova N.E., Alexandrov A.I., Ghazy E.S.M.O., Savin N.A., Gorelkin P.V., Erofeev A.S., Polshakov V.I. Antifungal Thiazolidines: Synthesis and Biological Evaluation of Mycosidine Congeners. Pharmaceuticals, 2022, 15, 5, 563-586. DOI: 10.3390/ph15050563тд1

     

  16. Treshchalin M.I., Polozkova V.A., Moiseenko E.I., Treshalina H.M., Shchekotikhin A.E., Pereverzeva E.R. Evaluation of Toxic Properties of New Glycopeptide Flavancin on Rats. Pharmaceuticals, 2022, 15, 661. DOI: 10.3390/ph15060661тл2

     

  17. A.N. Tevyashova, S.S. Efimova, A.I. Alexandrov, E.S.M.O. Ghazy, E.N. Bychkova, S.E. Solovieva, G.B. Zatonsky, N.E. Grammatikova, L.G. Dezhenkova, E.R. Pereverzeva, E.B. Isakova, O.S. Ostroumova, O.A. Omelchuk, V.V. Muravieva, M.M. Krotova, T.V. Priputnevich, A.E. Shchekotikhin, Semisynthetic Amides of Polyene Antibiotic Natamycin, ACS Infectious Diseases 2022, 2022, https://doi.org/10.1021/acsinfecdis.2c00237тл3
  18. A. Tevyashova, S. Efimova, A. Alexandrov, O. Omelchuk, E. Ghazy, E. Bychkova, G. Zatonsky, N. Grammatikova, L. Dezhenkova, S. Solovieva, O. Ostroumova, A. Shchekotikhin, Semisynthetic Amides of Amphotericin B and Nystatin A1: A Comparative Study of In Vitro Activity/Toxicity Ratio in Relation to Selectivity to Ergosterol Membranes, Antibiotics 2023, 12(1), 151; https://doi.org/10.3390/antibiotics12010151тл4